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Chemical Structure : AZD6280
Catalog No.: PC-62765Not For Human Use, Lab Use Only.
AZD6280 is a potent, α2/3 functionally selective, partial GABAA receptor modulator with pKi of 7.7.
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AZD6280 is a potent, α2/3 functionally selective, partial GABAA receptor modulator with pKi of 7.7; exerts neutral antagonism at the α1-subunit and partial efficacy at the α2,3-subunits over the α5-subunit, shows potential for the treatment of anxiety disorders.
Anxiety
Phase 1 Discontinued
| M.Wt | 366.421 | |
| Formula | C20H22N4O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Jucaite A, et al. Psychopharmacology (Berl). 2017 Feb;234(4):707-716.
2. Chen X, et al. J Clin Psychopharmacol. 2015 Feb;35(1):22-33.
3. Te Beek ET, et al. Clin Pharmacol Drug Dev. 2015 Mar;4(2):149-54.
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