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Chemical Structure : Daprodustat
CAS No.: 960539-70-2
Catalog No.: PC-45387Not For Human Use, Lab Use Only.
Daprodustat (GSK1278863) is a potent, orally active HIF-prolyl hydroxylase (PHD) inhibitor with IC50 of 3.5, 22.2 and 2.2 nM for PHD1, PHD2 and PHD3, respectively.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 25 mg | $198 | In stock | |
| 50 mg | $298 | In stock | |
| 100 mg | $498 | In stock | |
| 200 mg | Get quote | ||
| 1 g | Get quote |
Bulk size, bulk discount!
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| M.Wt | 393.4342 | |
| Formula | C19H27N3O6 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: < 6.8 mg/mL |
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| Chemical Name/SMILES |
Glycine, N-[(1,3-dicyclohexylhexahydro-2,4,6-trioxo-5-pyrimidinyl)carbonyl]- |
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1. Brigandi RA, et al. Am J Kidney Dis. 2016 Jun;67(6):861-71.
2. Hara K, et al. Drug Metab Pharmacokinet. 2015 Dec;30(6):410-8.
3. Johnson BM, et al. Clin Pharmacol Drug Dev. 2014 Mar;3(2):109-17.
4. Ariazi JL, et al. J Pharmacol Exp Ther. 2017 Dec;363(3):336-347.
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