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Chemical Structure : ENMD-2076 tartrate
CAS No.: 1291074-87-7
Catalog No.: PC-42765Not For Human Use, Lab Use Only.
A multitargeted kinase inhibitor with IC50s of 3/14/23/40 nM for Flt3/Aurora A/Src/VEGFR2.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $72 | In stock | |
| 50 mg | $116 | In stock | |
| 100 mg | $208 | In stock |
Bulk size, bulk discount!
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A multitargeted kinase inhibitor with IC50s of 3/14/23/40 nM for Flt3/Aurora A/Src/VEGFR2; also inhibits Aurora B, c-Kit, FGFR1 (IC50=100-350 nM); orally bioactive.
Liver Cancer
Phase 2 Clinical
| M.Wt | 525.5569 | |
| Formula | C25H31N7O6 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
4-Pyrimidinamine, 6-(4-methyl-1-piperazinyl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(1E)-2-phenylethenyl]- Tartrate |
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1. Tentler JJ, et al. Clin Cancer Res. 2010 Jun 1;16(11):2989-98.
2. Matulonis UA, et al. Eur J Cancer. 2013 Jan;49(1):121-31.
3. Fletcher GC, et al. Mol Cancer Ther. 2011 Jan;10(1):126-37.
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