You are here:Home-Chemical Inhibitors & Agonists-GPCR-5-HT Receptor-Eletriptan hydrobromide
Eletriptan hydrobromide

Chemical Structure : Eletriptan hydrobromide

CAS No.: 177834-92-3

Eletriptan hydrobromide (UK 116044 hydrobromide)

Catalog No.: PC-61867Not For Human Use, Lab Use Only.

Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.

Packing Price Stock Quantity
100 mg Get quote
250 mg Get quote
500 mg Get quote
1 g Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist; significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease; displays antimigraine activity.

Migraine

Approved

Physicochemical Properties

M.Wt 463.43
Formula C22H26N2O2S.HBr
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole hydrobromide

References

1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.

2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.

3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: