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Chemical Structure : GSK-2879552
CAS No.: 1401966-69-5
Catalog No.: PC-45495Not For Human Use, Lab Use Only.
GSK-2879552 is a potent, selective irreversible inhibitor of LSD1 with Ki app of 1.7 uM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $128 | In stock | |
| 25 mg | $198 | In stock | |
| 50 mg | $298 | In stock | |
| 100 mg | Get quote |
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GSK-2879552 is a potent, selective irreversible inhibitor of LSD1 with Ki app of 1.7 uM.
GSK-2879552 shows good selectivity against LSD2, MAO-A, MAO-B, D-amino acid oxidase and LoxL2.
GSK-2879552 exhibits growth inhibition (EC50=2-240 nM) in sensitive cell lines.
GSK-2879552 is orally bioavailable.
| M.Wt | 364.4806 | |
| Formula | C23H28N2O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
Benzoic acid, 4-[[4-[[[(1R,2S)-2-phenylcyclopropyl]amino]methyl]-1-piperidinyl]methyl]- |
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1. Mohammad HP, et al. Cancer Cell. 2015 Jul 13;28(1):57-69.
2. Huang M, et al. Cancer Lett. 2017 Jul 10;398:12-21.
3. Maes T, et al. Epigenomics. 2015;7(4):609-26.
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