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Chemical Structure : SJ830599
Catalog No.: PC-63255Not For Human Use, Lab Use Only.
SJ830599 is a modest selective BRD2-BD2 inhibitor with IC50 of 0.61 uM, 3.3-fold selectivity over BRD2-BD1.
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SJ830599 is a modest selective BRD2-BD2 inhibitor with IC50 of 0.61 uM, 3.3-fold selectivity over BRD2-BD1; demonstrates cytotoxicity against several pediatric cancer cell lines with EC50 values (HD-MB03 EC50=480 nM) comparable to BET inhibitor (BETi) clinical candidates.
| M.Wt | 356.422 | |
| Formula | C20H24N2O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Shadrick WR, et al. Bioorg Med Chem. 2018 Jan 1;26(1):25-36.
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