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Chemical Structure : VE-821
CAS No.: 1232410-49-9
Catalog No.: PC-44042Not For Human Use, Lab Use Only.
VE-821 (VE821) is a potent, selective and ATP-competitive inhibitor of ATR with Ki/IC50 of 13 nM/26 nM, respectively.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $58 | In stock | |
| 10 mg | $88 | In stock | |
| 25 mg | $128 | In stock | |
| 50 mg | $218 | In stock | |
| 100 mg | Get quote |
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VE-821 (VE821) is a potent, selective and ATP-competitive inhibitor of ATR with Ki/IC50 of 13 nM/26 nM, respectively.
VE-821 shows excellent selectivity for ATR over the related PIKKs ATM, DNA-PK, mTOR and PI3K.
| M.Wt | 368.4096 | |
| Formula | C18H16N4O3S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
2-Pyrazinecarboxamide, 3-amino-6-[4-(methylsulfonyl)phenyl]-N-phenyl- |
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1. Reaper PM, et al. Nat Chem Biol, 2011, 7(7), 428-430.
2. Charrier JD, et al. J Med Chem, 2011, 54(7), 2320-2330.
3. Prevo R, et al. Cancer Biol Ther. 2012 Sep;13(11):1072-81.
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