| Cat. No. |
Product Name |
Information |
| PC-70072 |
ST1535
A2AR antagonist
|
ST1535 is a potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM. |
| PC-45641 |
ZM241385
A2A receptor inhibitor
|
ZM241385 is a potent, non-xanthine A2A-selective adenosine receptor antagonist with rat PC12 binding pIC50 of 9.52. |
| PC-45642 |
SCH 58261
A2AR antagonist
|
SCH 58261 is a potent and selective, competitive A2A adenosine receptor antagonist with Ki of 2.3 nM and 2.0 nM in rat and bovine brain, respectively. |
| PC-42064 |
eN-IN-1
CD73 inhibitor
|
An α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 29 nM for rat recombinant eN. |
| PC-42043 |
CI-947
Adenosine receptor agonist
|
An orally active adenosine receptor agonist that can induce acute cardiovascular toxicity and coronary vascular injury in vivo.. |
| PC-45566 |
N6-Cyclohexyladenosine
A1AR agonist
|
N6-Cyclohexyladenosine is an adenosine A1 receptor agonist (EC50= 8.2 nM). |
| PC-44125 |
Capadenoson
A1AR agonist
|
Capadenoson (BAY68-4986) is a selective agonist of adenosine-A1 receptor (A1AR). |
| PC-42771 |
Tozadenant
A2AR antagonist
|
Tozadenant (SYN115) is a potent, selective adenosine 2A receptor (A2AR) antagonist with Ki of 11.5 nM. |
| PC-45585 |
GR-79236
A1AR agonist
|
GR-79236 is a potent and selective Adenosine A1 receptor agonist with Ki of 3.1 nM. |
| PC-42717 |
Vipadenant
A2AR antagonist
|
Vipadenant (BIIB014) is a potent and selective A2A adenosine receptor antagonist with Ki of 1.3 nM. |
| PC-42729 |
Preladenant
A2AR antagonist
|
Preladenant (SCH420814) is a potent and highly selective adenosine A2A receptor competitive antagonist with Ki of 1.1 nM. |
| PC-42728 |
Istradefylline
A2AR antagonist
|
Istradefylline (KW6002) is a potent and highly selective A2A receptor antagonist with Ki of 2.2 nM. |
