| Cat. No. |
Product Name |
Information |
| PC-20307 |
BAY-6096
Adrenergic α2B inhibitor
|
BAY-6096 (BAY6096) is a potent, selective, and highly water-soluble adrenergic α2B antagonist with IC50 of 14 nM. |
| PC-49058 |
AS408
β2AR modulator
|
AS408 is a negative allosteric modulator of the β2-adrenergic receptor (β2AR) for both G-protein activation and arrestin recruitment (pKB=6.8, [35S]GTPγS binding assays), binds to a pocket formed by the membrane-facing surface of TM3 and TM5. |
| PC-47093 |
Tasipimidine
α2A adrenoceptor agonist
|
Tasipimidine is a potent, selective and orally active human α2A-adrenoceptor agonist with pEC50 of 7.57, >100-fold selectivity over α2B-and α2C-adrenoceptors and the rodent α2D-adrenoceptor. |
| PC-36084 |
Olodaterol hydrochloride
|
Olodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2. |
| PC-35360 |
AGN192836
α2AR agonist
|
AGN192836 (AGN 192836) is a potent, selective α2 adrenergic (alpha 2-adrenoceptor, α2AR) agonist with EC50 of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. |
| PC-35028 |
BI 167107
β2AR agonist
|
BI 167107 is a highly potent agonist of the β2 adrenergic receptor (β2AR) and β1AR (IC50=3.2 nM) and shows some activity as α1A antagonist (IC50 = 32 nM). |
| PC-62018 |
BRL 37344 sodium
β3 adrenoceptor agonist
|
BRL 37344 sodium (BRL 37344A) is a potent and selective β3 adrenoceptor agonist with Ki of 287 nM. |
| PC-62017 |
CL 316243
β3 adrenoceptor agonist
|
CL 316243 (BTA 243) is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM. |
| PC-62016 |
CL 316243 disodium
β3 adrenoceptor agonist
|
CL 316243 is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM. |
| PC-61778 |
Xamoterol hemifumarate
β1AR agonist
|
Xamoterol (ICI 118587) is a third-generation adrenergic β1 adrenergic receptor partial agonist that acts as a cardiac stimulant.. |
| PC-60734 |
MK-4618
β3 adrenergic receptor agonist
|
MK-4618 (Vibegron, KRP-114V, RVT-901) is a potent and selective full β3 adrenergic receptor agonist with EC50 of 1.1 nM. |
| PC-21223 |
ZD7114
beta-adrenoceptor agonist
|
ZD7114 (ICI D7114) is a potent, selective beta-adrenoceptor agonist, selectively stimulates brown fat and increases whole-body oxygen consumption. |
