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Cat. No. Product Name Information
PC-21190

Bestatin

CD13 inhibitor

Ubenimex (Bestatin) is a natural, broad-spectrum, and competitive CD13 (Aminopeptidase N)/APN and leukotriene A4 hydrolase inhibitor with anticancer effects.
PC-49177

BDM88951

ERAP2 inhibitor

BDM88951 (BDM 88951) is a highly potent, selective inhibitor of endoplasmic reticulum aminopeptidase 2 (ERAP2) with IC50 of 19 nM.
PC-73107

M8891

MetAP-2 inhibitor

M8891 (M 8891) is an orally bioavailable, potent, and reversible methionine aminopeptidase 2 (MetAP2) inhibitor with IC50 of 54 nM, Ki of 4.33 nM.
PC-72623

ST-115

Aminopeptidase P2 inhibitor

ST-115 (ST115) is a potent and specific inhibitor of aminopeptidase P2 ((XPNPEP2, APP2) with IC50 of 3.7 nM.
PC-72273

IRAP-IN-1

IRAP inhibitor

IRAP-IN-1 is a selective insulin-regulated aminopeptidase (IRAP) inhibitor with IC50 of 32 nM, >25-fold selectivity over ERAP1 and ERAP2.
PC-72271

DG013A

ERAP1 inhibitor

DG013A (DG 013A) is tripeptide mimetic chemical probe (inhibitor) of ERAP1 with IC50 of 0.19 uM, 15-fold selectivity over ERAP2, potently inhibits aminopeptidase N (APN) with IC50 of 3.7 nM.
PC-38334

CARD8 activator CQ31

PEPD/XPNPEP1 inhibitor

CARD8 activator CQ31 is a small molecule that selectively activates CARD8, inhibits the M24B aminopeptidases prolidase (PEPD) and Xaa-Pro aminopeptidase 1 (XPNPEP1), leading to the accumulation of proline-containing peptides that inhibit DPP8/9 and thereby activate CARD8.
PC-35112

TP-004

MetAP-2 inhibitor

TP-004 is a potent, selective and reversible inhibitor of methionine aminopeptidase 2 (MetAP2) with IC50 of 6 nM.
PC-63347

A-800141

MetAP2 inhibitor

A-800141 is a potent, highly specific, orally bioavailable MetAP2 inhibitor with IC50 of 12 nM, shows no inhibition for MetAP1 (IC50>30 uM).
PC-63319

PPI-2458

MetAP-2 inhibitor

PPI-2458 is potent, specific, irreversible methionine aminopeptidase-2 (MetAP-2) inhibitor with IC50 of 0.2 nM, inhibits growth inhibition of HFLS-RA and HUVEC with IC50 of 0.04 nM.
PC-63318

A-357300

MetAP2 inhibitor

A-357300 is a potent, selective, reversible MetAP2 inhibitor with IC50 of 0.12 uM, does not inhibit MetAP1 or leucine aminopeptidases at 10 uM.
PC-63317

A-832234

MetAP-2 inhibitor

A-832234 is a potent, selective, reversible MetAP2 inhibitor with IC50 of 19 nM..

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