(R)-PG648 | D3R antagonist | Probechem Biochemicals

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Chemical Structure : (R)-PG648

(R)-PG648 (Compound R-22)

Catalog No.: PC-27836Not For Human Use, Lab Use Only.

(R)-PG648 (Compound R-22) is a potent, selective dopamine D3 receptor (D3R) antagonist with Ki of 1.12 nM, 400-fold more selective for D3R over D2R.

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Biological Activity

(R)-PG648 (Compound R-22) is a potent, selective dopamine D3 receptor (D3R) antagonist with Ki of 1.12 nM, 400-fold more selective for D3R over D2R.

Physicochemical Properties

M.Wt	461.39
Formula	C23H26Cl2N4O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-3-hydroxybutyl)1H-indole-2-carboxamide

References

1. Ellen Y T Chien, et al. Science. 2010 Nov 19;330(6007):1091-5.

2. Vivek Kumar, et al. ACS Med Chem Lett. 2014 Mar 24;5(6):647-51.

3. Newman AH, et al. J. Med. Chem. 2009;52:2559.

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(R)-PG648 (Compound R-22)

Biological Activity

Physicochemical Properties

References

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