| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-62481 |
PS 210
|
1221962-86-2 |
PS 210 is a potent, specific activator of PDK1 that target the PIF-binding pocket of PDK1, does not alter the activity of any of the 121 kinases (S6K, PKB/Akt or GSK3).. |
| PC-60606 |
OSU-03013
|
742112-34-1 |
OSU-03013 (OSU 03013, OSU03013) is a novel potent, orally active 3-phosphoinositide-dependent kinase-1 (PDK-1) with IC50 of 2 uM. |
| PC-60605 |
OSU-03012
|
742112-33-0 |
OSU-03012 (AR-12) is a novel potent, orally active 3-phosphoinositide-dependent kinase-1 (PDK-1) with IC50 of 5 uM. |
| PC-42781 |
BX-912
|
702674-56-4 |
BX-912 (BX912) is a potent, selective and ATP-competitive inhibitor of PDK1 with IC50 of 26 nM. |
| PC-42629 |
BX795
|
702675-74-9 |
BX795 is a potent and relatively specific PDK1 inhibitor with IC50 of 6 nM. |
| PC-49261 |
GSK2334470
|
1227911-45-6 |
GSK2334470 (GSK 2334470) is a potent, highly specific inhibitor of PDK1 with IC50 of 10 nM, does not inhibit 93 other protein kinases including 13 AGC-kinases most related to PDK1 at 5 uM. |
| PC-73258 |
PDK-1 agonist PS48
|
1180676-32-7 |
PDK-1 agonist PS48 is a small molecule allosteric PDK-1 agonist, PS48 is active at 10 nM to 1 μM in restoring normal insulin-dependent Akt activation and in mitigating Aβi peptide toxicity. |
