| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-38860 |
IK-175
|
2247950-42-9 |
IK-175 is a potent, selective and orally active aryl hydrocarbon receptor (AHR) antagonist with IC50 of 91 nM in human HepG2 cells expressing an AHR-dependent DRE-luciferase reporter and stimulated with 80 nM of the AHR agonist VAF347. |
| PC-61627 |
FICZ
|
172922-91-7 |
FICZ is a high affinity aryl hydrocarbon receptor (AhR) agonist with Kd of 70 pM. |
| PC-60776 |
5F 203
|
260443-89-8 |
5F 203 (NSC 703786) is a potent, selective antitumour agent through activation the aryl hydrocarbon receptor (AhR) pathway. |
| PC-45600 |
ITE
|
448906-42-1 |
A endogenous ligand, potent aryl hydrocarbon receptor (AhR) agonist in vitro. |
| PC-38597 |
KYN-101
|
2247950-73-6 |
KYN-101 (KYN101) is a potent, selective synthetic antagonist of aryl hydrocarbon receptor (AHR) with IC50 of 22 nM in human HepG2 DRE-luciferase reporter assay and 23 nM in murine Hepa1 Cyp-luc assay. |
| PC-38513 |
SGA360
|
680611-86-3 |
SGA360 is a high-affinity, selective modulator of aryl hydrocarbon receptor (AhR), competitively binds to AhR (IC50 =3 uM) and represses serum amyloid A 1 (SAA1) gene expression induced by IL-1β in Huh7 cells. |
| PC-38065 |
BAY 2416964
|
2242464-44-2 |
BAY 2416964 is a potent and orally active aryl hydrocarbon receptor (AHR) antagonist with IC50 of 341 nM.. |
