| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-72402 |
M3258
|
2285330-15-4 |
M3258 (M 3258) is a potent, reversible, highly selective and orally acitve LMP7 inhibitor with cellular IC50 of 4.1 nM. |
| PC-43439 |
MG-132
|
133407-82-6 |
MG-132 (Z-Leu-leu-leu-al, Zlllal) is a potent, reversible, and cell-permeable proteasome inhibitor with IC50 of 0.1 and 1.2 μM for the inhibition of proteasome and calpain, respectively. |
| PC-61352 |
O-phenanthroline
|
66-71-7 |
A selective inhibitor of 26S proteasome subunit Rpn11 with IC50 of 10±2 uM. |
| PC-61193 |
CSN5i-3
|
2375740-98-8 |
CSN5i-3 (CSN5 inhibitor 3) is a potent, selective and orally available inhibitor of CSN5 with IC50 of 5.8 nM, the proteolytic subunit of COP9 signalosome (CSN). |
| PC-61132 |
Rpn11 inhibitor 35
|
2084868-04-0 |
Rpn11 inhibitor 35 is a potent, small molecule inhibitor of the proteasome subunit Rpn11 with IC50 of 400 nM,100-fold selectivity over Csn5 and 10-fold selectivity over AMSH. |
| PC-60969 |
NC-001
|
1237540-68-9 |
NC-001 (NC 001, NC001, az-NC-001) is a potent, specific, cell-permeable inhibitor of immunoproteasome caspase-like sites (β1i and β1), does not correlate with inhibition of chymotrypsin-like sites.. |
| PC-60968 |
ML 604440
|
1140517-08-3 |
ML 604440 (ML604440, ML-604440) is a potent, specific and cell permeable proteasome β1i (LMP2) subunit inhibitor. |
