| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-62770 |
MRK-623
|
461449-78-5 |
MRK-623 is a potent, α2/α3 subunit functionally selectiviie GABAA receptor agonist.. |
| PC-62098 |
LAU159
|
2055050-87-6 |
LAU159 is a potent, functionally selective positive modulator of α6β3γ2 GABAA receptor.. |
| PC-62089 |
PF-06372865
|
1614245-70-3 |
PF-06372865 (Darigabat) is a novel potent, α2/3 functionally selective GABAA receptor positive allosteric modulator. |
| PC-61895 |
Alprazolam
|
28981-97-7 |
Alprazolam (D-65MT, U 31889) is a triazolobenzodiazepine agent with anxiolytic, sedative-hypnotic and anticonvulsant activities. |
| PC-42117 |
MRK-016
|
342652-67-9 |
MRK-016 (MRK016) is a potent, functionally selective, CNS-penetrating and orally bioavailable inverse agonist of benzodiazepine site of GABAA α5 receptor with Ki of 0.8-1.5 nM for α1-, α2-, α3-, andα5-containing GABAA receptors. |
| PC-49725 |
KRM-II-81
|
2014348-91-3 |
KRM-II-81 is a selective α2/α3 subtype GABAA receptor ligand (positive allosteric modulator) with EC50 of 937 nM for α3β3γ2 GABAAR, with no potency against α1β3γ2. |
| PC-49338 |
EVT-201
|
308239-86-3 |
EVT-201 (Dimdazenil, EVT 201) is a partial positive allosteric GABA(A) receptor modulator with potential for the treatment of insomnia. |
