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Cat. No. Product Name Information
PC-20307

BAY-6096

Adrenergic α2B inhibitor

BAY-6096 (BAY6096) is a potent, selective, and highly water-soluble adrenergic α2B antagonist with IC50 of 14 nM.
PC-49058

AS408

β2AR modulator

AS408 is a negative allosteric modulator of the β2-adrenergic receptor (β2AR) for both G-protein activation and arrestin recruitment (pKB=6.8, [35S]GTPγS binding assays), binds to a pocket formed by the membrane-facing surface of TM3 and TM5.
PC-47093

Tasipimidine

α2A adrenoceptor agonist

Tasipimidine is a potent, selective and orally active human α2A-adrenoceptor agonist with pEC50 of 7.57, >100-fold selectivity over α2B-and α2C-adrenoceptors and the rodent α2D-adrenoceptor.
PC-36084

Olodaterol hydrochloride

Olodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2.
PC-35360

AGN192836

α2AR agonist

AGN192836 (AGN 192836) is a potent, selective α2 adrenergic (alpha 2-adrenoceptor, α2AR) agonist with EC50 of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively.
PC-35028

BI 167107

β2AR agonist

BI 167107 is a highly potent agonist of the β2 adrenergic receptor (β2AR) and β1AR (IC50=3.2 nM) and shows some activity as α1A antagonist (IC50 = 32 nM).
PC-43176

Midodrine

α1-adrenoceptor agonist

Midodrine is a selective α1-adrenoceptor agonist that acts as a vasopressor/antihypotensive agent for the treatment of dysautonomia and orthostatic hypotension.
PC-43012

Atipamezole

α2 adrenoceptor agonist

Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM.
PC-62018

BRL 37344 sodium

β3 adrenoceptor agonist

BRL 37344 sodium (BRL 37344A) is a potent and selective β3 adrenoceptor agonist with Ki of 287 nM.
PC-62017

CL 316243

β3 adrenoceptor agonist

CL 316243 (BTA 243) is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM.
PC-62016

CL 316243 disodium

β3 adrenoceptor agonist

CL 316243 is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM.
PC-62004

Milveterol

β2 adrenoceptor agonist

Milveterol (GSK 159797) is a potent, selective long-acting β2 adrenoceptor agonist with pEC50 of 10.2 in cell-based assays, displays good β2/β1 selectivity (>300-fold).

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