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Cat. No. Product Name Information
PC-38542

Takeda103A

GRK2 inhibitor

Takeda103A is a potent, selective GRK2 inhibitor with IC50 of 0.02 uM, 450-fold selectivity over GRK5.
PC-72421

GRK6 inhibitor 18

GRK6 inhibitor

GRK6 inhibitor 18 is a potent, and selective GRK6 inhibitor with IC50 of 8 nM.
PC-60588

CCG 258001

GRK2 inhibitor

CCG 258001 is a potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM.
PC-60587

CCG 224061

GRK2 inhibitor

A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 66 nM.
PC-60586

CCG 258748

GRK2 inhibitor

CCG 258748 is a potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.
PC-60585

Compound 101

GRK2/3 inhibitor

Compound 101 (GRK2 inhibitor 101, Takeda compound 101, Cmpd101) is a novel membrane-permeable, small-molecule inhibitor of GRK2 and GRK3 with IC50 of 18 nM and 5.4 nM, respectively.
PC-60353

GRK2-IN-115h hydrochloride

GRK2 inhibitor

GRK2-IN-115h hydrochloride is a highly potent and selective GRK2 inhibitor with IC50 of 18 nM.
PC-70119

CCG-224406

GRK2 inhibitor

CCG-224406 (CCG224406) is a highly selective and potent GRK2 (G protein-coupled receptor kinase 2) inhibitor with IC50 of 130 nM.M.
PC-45591

CCG215022

GRK inhibitor

CCG-215022 (CCG215022) is a potent and selective pan GRK (G protein-coupled receptor kinase) inhibitor with IC50 of 0.15/0.38/3.9 uM for GRK2/5/1 respectively.
PC-45590

GSK180736A

GRK2 inhibitor

GSK180736A is a highly selective and potent GRK2 inhibitor with IC50 of 0.77 uM.
PC-21461

GRL018-21

GRK5 inhibitor

GRL018-21 is a highly selective, potent, and non-covalent GRK5 inhibitor with IC50 of 10 nM, >100,000-fold selectivity over GRK2.

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