| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-63122 |
YKL 06-061
|
2172617-15-9 |
YKL 06-061 is a potent, selective, second-generation salt-inducible kinase (SIK) inhibitor with IC50 of 6.56/1.77/20.5 nM for SIK1/2/3, respectively. |
| PC-61766 |
ARN-3236
|
1613710-01-2 |
ARN-3236 is a novel potent, selective, and orally active SIK2 inhibitor with IC50 of <1 nM. |
| PC-42327 |
YKL-05-099
|
1936529-65-5 |
YKL-05-099 (YKL 05-099) is a novel potent, selective pan-SIK inhibitor with IC50 of 10, 40 and 30 nM for SIK1, 2 and 3, respectively. |
| PC-49563 |
SK-124
|
2760404-50-8 |
SK-124 (SK124) is a potent, selective, orally active SIK2/SIK3 inhibitor with IC50 of 8.8/11.3 nM in cell-based NanoBRET assays, 15-fold selectivity versus SIK1. |
| PC-72723 |
MRIA9
|
2750707-05-0 |
MRIA9 is a potent, selective dual SIK/PAK inhibitor, inhibits SIK1/2/3 with cellular IC50 of 586/180/127 nM, respectively. |
| PC-63124 |
rac Pterosin B
|
60657-37-6 |
rac Pterosin B is a potent and specific SIK3 signaling inhibitor that suppresses SIK3 downstream cascades by up-regulating the phosphorylation levels in the SIK3 C-terminal regulatory domain. |
| PC-63123 |
Pterosin B
|
34175-96-7 |
Pterosin B is a potent and specific SIK3 signaling inhibitor that suppresses SIK3 downstream cascades by up-regulating the phosphorylation levels in the SIK3 C-terminal regulatory domain. |
