| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-36169 |
FB23-2
|
2243736-45-8 |
FB23-2 is a potent, selective inhibitor of the mRNA N 6-methyladenosine (m 6A) demethylase FTO, directly bind to FTO, inhibits FTO demethylation of m6 A in RNA in vitro with IC50 of 2.6 uM. |
| PC-35471 |
Vafidemstat
|
1357362-02-7 |
Vafidemstat (ORY-2001, ORY2001) is a potent, selective, brain penetrant dual lysine-specific histone demethylase (LSD1, KDM1A)/MAO-B inhibitor with IC50 of 105 nM (KDM1A) and 58 nM (MAO-B). |
| PC-43206 |
ORY-1001 trans and cis isomers
|
1431326-61-2 |
ORY-1001 (RG-6016) is a highly potent, selective inhibitor of lysine-specific demethylase KDM1A (LSD1) with IC50 of 18 nM, displays high selectivity for KDM1A over other FAD-containing monoamine oxidases. |
| PC-62293 |
GS-5801
|
1596348-32-1 |
KDM5-C70 (GS-5801) is a cell-permeable derivative of KDM5-C49 (GS-080), potent, selective and cell permeable KDM5 inhibitor with IC50 of 0.3, 0.3 and 0.58 uM for KDM5A, B and C, respectively. |
| PC-61739 |
QC-6352
|
1851373-36-8 |
QC-6352 is a potent and selective KDM4 family inhibitor with IC50 of 104, 56, 35, and 104 nM for KDM4A, KDM4B, KDM4C, and KDM4D, respectively. |
| PC-61398 |
Seclidemstat
|
1423715-37-0 |
Seclidemstat (SP-2577, SP2577) is a potent, selective LSD1 inhibitor with IC50 of 127 nM. |
| PC-70332 |
SD-70
|
332173-89-4 |
SD-70 is a small molecule tumor translocation inhibitor that inhibits the prostate cancer cell transcriptional program, in part by inhibition of the demethylase KDM4C (IC50=30 uM). |
