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Cat. No. Product Name CAS No. Information
PC-73454

Vicasinabin

1433361-02-4 Vicasinabin (RG7774, RG-7774) is a potent, selective agonist of cannabinoid receptor 2 (CB2) with cAMP EC50 of 1 nM (hCB2), >800-fold selectivity over CB1 receptor.
PC-43210

CB1-IN-4

1429239-98-4 DBPR211 (BPRCB1184, CB1-IN-4) is a potent, selective, peripherally restricted cannabinoid-1 (CB1) receptor antagonist with Ki of 0.3 nM, EC50 of 3.0 nM.
PC-60146

APD-371

1268881-20-4 APD-371 (APD371, Olorinab) is a potent, selective and orally available CB2 agonist with EC50 of 6.2 nM.
PC-60086

AM-6538

1245626-00-9 AM-6538 (AM6538) is a potent, selective cannabinoid receptor CB1 antagonist with Ki of 5.1 nM..
PC-49218

S-777469

885496-53-7 S-777469 (S777469) is a potent, selective, orally available cannabinoid receptor 2 (CB2) receptor agonist with Ki value of 32 nM (hCB2), >100-fold selectivity over CB1.
PC-47097

LY2828360

1231220-79-3 LY2828360 is a potent CB2 receptor agonist with similar affinity for human and rat CB2 receptors with Ki of 40.3 nM and 36.7 nM, respectively, shows EC50 of 20.1 nM in [35S]-GTPγS assays.
PC-38638

JM-00266

2090325-46-3 JM-00266 is a novel non-brain penetrant cannabinoid receptor 1 (CB1R) inverse agonist.

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