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Chemical Structure : ACT-1016-0707
Catalog No.: PC-21751Not For Human Use, Lab Use Only.
ACT-1016-0707 is a potent, selective, and orally active lysophosphatidic acid receptor subtype 1 receptor (LPA1 receptor, LPAR1) antagonist with IC50 of 3.1 nM, highly selective over LPAR2 or LPAR3.
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ACT-1016-0707 is a potent, selective, and orally active lysophosphatidic acid receptor subtype 1 receptor (LPA1 receptor, LPAR1) antagonist with IC50 of 3.1 nM, highly selective over LPAR2 or LPAR3.
ACT-1016-0707 suppressed the LPA-induced vascular leakage at a p.o. dose of 30 mg/kg.
| M.Wt | 438.93 | |
| Formula | C19H23ClN4O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Lescop C, et al. J Med Chem. 2024 Feb 13. doi: 10.1021/acs.jmedchem.3c01827.
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