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Chemical Structure : ACT-281959
Catalog No.: PC-35578Not For Human Use, Lab Use Only.
ACT-281959 (ACT281959) is the prodrug of ACT-246475, which is a potent, selective, reversible P2Y12 receptor antagonist with binding IC50 of 1.0 nM.
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ACT-281959 (ACT281959) is the prodrug of ACT-246475, which is a potent, selective, reversible P2Y12 receptor antagonist with binding IC50 of 1.0 nM; ACT-281959 is orally acitve, shows efficacy in the rat ferric chloride thrombosis model.
| M.Wt | 850.86 | |
| Formula | C38H55N6O14P | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Caroff E, et al. J Med Chem. 2015 Dec 10;58(23):9133-53.
2. Rey M, et al. Pharmacol Res Perspect. 2017 Oct;5(5).
3. Juif PE, et al. J Clin Pharmacol. 2018 Aug 8. doi: 10.1002/jcph.1296.
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