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Chemical Structure : AR NTD inhibitor 16
CAS No.: 3016437-05-8
Catalog No.: PC-21578Not For Human Use, Lab Use Only.
AR NTD inhibitor 16 is a small molecule inhibitor of androgen receptor N-terminal domain (AR NTD) with IC50 of 0.12 uM in VCaP cell-based GRE2-luciferase reporter gene assays.
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AR NTD inhibitor 16 is a small molecule inhibitor of androgen receptor N-terminal domain (AR NTD) with IC50 of 0.12 uM in VCaP cell-based GRE2-luciferase reporter gene assays.
AR NTD inhibitor 16 is more potent than known AR-NTD AF1 binder EPI-001 (IC50=37.4 μM).
AR NTD inhibitor 16 is a tool compound to investigate the pharmacology and engagement of the AR NTD.
| M.Wt | 297.38 | |
| Formula | C16H15N3OS | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
Benzamide, 3-(1-methyl-1H-indazol-5-yl)-4-(methylthio)- |
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1. Martyn C Henry, et al. ACS Med Chem Lett. 2023 Nov 17;14(12):1800-1806.
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