Chemical Structure : AZD1283
CAS No.: 919351-41-0
Catalog No.: PC-20648Not For Human Use, Lab Use Only.
AZD1283 (AZD-1283) is a potent, selective P2Y12 receptor antagonist with binding IC50 of 11 nM, and IC50 of 3.2 uM in washed platelet assay (WPA).
Packing | Price | Stock | Quantity |
---|---|---|---|
5 mg | $198 | In stock | |
25 mg | $498 | In stock | |
100 mg | Get quote | ||
200 mg | Get quote | ||
1 g | Get quote |
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
AZD1283 (AZD-1283) is a potent, selective P2Y12 receptor antagonist with binding IC50 of 11 nM, and IC50 of 3.2 uM in washed platelet assay (WPA).
AZD1283 dose-dependently induced increases in blood flow and inhibition of ADP-induced platelet aggregation with antithrombotic ED50 values of 3.0 μg/kg/min.
M.Wt | 470.54 | |
Formula | C23H26N4O5S | |
Appearance | Solid | |
Storage |
|
|
Solubility |
10 mM in DMSO |
|
Chemical Name/SMILES |
CC1=C(C(OCC)=O)C=C(C#N)C(N2CCC(C(NS(=O)(CC3=CC=CC=C3)=O)=O)CC2)=N1 |
1. Kong D, et al. J Med Chem. 2019 Mar 28;62(6):3088-3106.
2. Bach P, et al. J Med Chem. 2013 Sep 12;56(17):7015-24.
3. Zhang K, et al. Nature. 2014 May 1;509(7498):115-8.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright