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Chemical Structure : Acebilustat
CAS No.: 943764-99-6
Catalog No.: PC-45393Not For Human Use, Lab Use Only.
Acebilustat (CTX-4430, EP-501) is a potent and selective leukotriene A4 hydrolase (LTA4H) inhibitor with IC50 of 64 nM for inhibition of LTB4 production in human whole blood.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 25 mg | $188 | In stock | |
| 50 mg | $298 | In stock | |
| 100 mg | $488 | In stock | |
| 200 mg | Get quote | ||
| 1 g | Get quote |
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Acebilustat (CTX-4430, EP-501) is a potent and selective leukotriene A4 hydrolase (LTA4H) inhibitor with IC50 of 64 nM for inhibition of LTB4 production in human whole blood.
Acebilustat (CTX-4430, EP-501) a new once‐daily oral antiinflammatory drug in development for treatment of cystic fibrosis (CF) and other diseases.
| M.Wt | 481.5424 | |
| Formula | C29H27N3O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO; Methanol: ≥ 32 mg/mL |
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| Chemical Name/SMILES |
Benzoic acid, 4-[[(1S,4S)-5-[[4-[4-(2-oxazolyl)phenoxy]phenyl]methyl]-2,5-diazabicyclo[2.2.1]hept-2-yl]methyl]- |
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1. Elborn JS, et al. Clin Transl Sci. 2017 Jan;10(1):20-27.
2. Elborn JS, et al. Clin Transl Sci. 2017 Jan;10(1):28-34.
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