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Chemical Structure : Aprocitentan
Catalog No.: PC-60030Not For Human Use, Lab Use Only.
A major and pharmacologically active metabolite of Macitentan, an orally active, dual endothelin receptor antagonist.
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A major and pharmacologically active metabolite of Macitentan, an orally active, dual endothelin receptor antagonist; inhibits ET-1 and ET-2-induced contractions in functional assays.
| M.Wt | 546.194 | |
| Formula | C16H14Br2N6O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Iglarz M, et al. J Pharmacol Exp Ther. 2008 Dec;327(3):736-45.
2. Kummer O, et al. Eur J Pharm Sci. 2009 Nov 5;38(4):384-8.
3. Sidharta PN, et al. Eur J Clin Pharmacol. 2011 Oct;67(10):977-84.
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