You are here:Home-Chemical Inhibitors & Agonists-GPCR-Luteinizing Hormone Receptor (LHR)-BAY-899
BAY-899

Chemical Structure : BAY-899

CAS No.: 2471967-92-5

BAY-899 (BAY899)

Catalog No.: PC-72912Not For Human Use, Lab Use Only.

BAY-899 (BAY899) is a highly potent, selective luteinizing hormone receptor (LH-R) inhibitor with IC50 of 185 nM and 46 nM for hLH-R and rLH-R, respectively.

Packing Price Stock Quantity
5 mg $148 In stock
10 mg $218 In stock
25 mg $358 In stock
100 mg Get quote
250 mg Get quote
1 g Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

BAY-899 (BAY899) is a highly potent, selective luteinizing hormone receptor (LH-R) inhibitor with IC50 of 185 nM and 46 nM for hLH-R and rLH-R, respectively.
BAY-899 reduces sex hormone levels in vivo.
BAY-899 is a valuable tool compound to study hLH-R signaling in vitro and to interfere with the production of sex hormones in vivo.

Physicochemical Properties

M.Wt 459.457
Formula C25H19F2N5O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(5S)-N-[2-(4-Fluorophenoxy)pyrimidin-5-yl]-5-(4-fluorophenyl)-7,8-dihydro-1,6-naphthyridine-6(5H)-carboxamide

References

1. Lars Wortmann, et al. J Med Chem. 2019 Nov 27;62(22):10321-10341.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: