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Chemical Structure : Bay 59-3074
CAS No.: 406205-74-1
Catalog No.: PC-42171Not For Human Use, Lab Use Only.
Bay 59-3074 is a potent, selective cannabinoid CB1/CB2 receptor partial agonist with Ki of 48.3, and 45.5 nM for human CB1 and human CB2 receptors, respectively.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $88 | In stock | |
| 25 mg | $148 | In stock | |
| 50 mg | $238 | In stock | |
| 100 mg | Get quote |
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Bay 59-3074 is a potent, selective cannabinoid CB1/CB2 receptor partial agonist with Ki of 48.3, and 45.5 nM for human CB1 and human CB2 receptors, respectively.
Bay 59-3074 displays antihyperalgesic and antiallodynic effects against thermal or mechanical stimuli in rat models of chronic neuropathic; orally acitve.
| M.Wt | 453.3555 | |
| Formula | C18H13F6NO4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 34 mg/mL |
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| Chemical Name/SMILES |
1-Butanesulfonic acid, 4,4,4-trifluoro-, 3-[2-cyano-3-(trifluoromethyl)phenoxy]phenyl ester |
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1. De Vry J, et al. J Pharmacol Exp Ther. 2004 Aug;310(2):620-32.
2. De Vry J, et al. Eur J Pharmacol. 2004 Nov 28;505(1-3):127-33.
3. Teng H, et al. Bioorg Med Chem Lett. 2011 Oct 1;21(19):5999-6002.
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