You are here:Home-Chemical Inhibitors & Agonists-Membrane Transporter/Ion Channel-BCRP-Brevianamide F
Brevianamide F

Chemical Structure : Brevianamide F

CAS No.: 38136-70-8

Brevianamide F (Cyclo(L-Pro-L-Trp))

Catalog No.: PC-42127Not For Human Use, Lab Use Only.

A naturally occurring 2,5-diketopiperazine that possess interesting breast cancer resistance protein (BCRP) inhibitory activity..

Packing Price Stock Quantity
10 mg $120 In stock
50 mg $360 In stock
100 mg $560 In stock

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

A naturally occurring 2,5-diketopiperazine that possess interesting breast cancer resistance protein (BCRP) inhibitory activity.; also shows agonism towards Ca(2+)-channel activity at 100 uM, and has potentiation for use in the treatment of cardiovascular dysfunction.

Physicochemical Properties

M.Wt 283.3251
Formula C16H17N3O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

Pyrrolo[1,2-a]pyrazine-1,4-dione, hexahydro-3-(1H-indol-3-ylmethyl)-, (3S,8aS)-

References

1. Jamie H, et al. J Pharm Pharmacol. 2002 Dec;54(12):1659-65.

2. Wauters I, et al. J Org Chem. 2015 Aug 21;80(16):8046-54.

3. Wollinsky B, et al. Org Biomol Chem. 2012 Dec 14;10(46):9262-70.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: