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Chemical Structure : CCG-224406
Catalog No.: PC-70119Not For Human Use, Lab Use Only.
A highly selective and potent GRK2 (G protein-coupled receptor kinase 2) inhibitor with IC50 of 130 nM.
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A highly selective and potent GRK2 (G protein-coupled receptor kinase 2) inhibitor with IC50 of 130 nM; displays >700-fold selectivity over other GRK subfamilies, and no detectable inhibition of ROCK1.
| M.Wt | 558.57 | |
| Formula | C29H27FN6O5 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Waldschmidt HV, et al. J Med Chem. 2016 Apr 28;59(8):3793-807.
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