CDK12-IN-3

Chemical Structure : CDK12-IN-3

CAS No.: 2220184-50-7

Catalog No.: PC-28041Not For Human Use, Lab Use Only.

CDK12-IN-3 is a potent, selective, noncovalent CDK12 inhibitor with IC50 of 491 nM, inhibits phosphorylation of Ser2 on the C-terminal repeat domain of RNA polymerase II.

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10 mg	$458	In stock
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Biological Activity

CDK12-IN-3 is a potent, selective, noncovalent CDK12 inhibitor with IC50 of 491 nM, inhibits phosphorylation of Ser2 on the C-terminal repeat domain of RNA polymerase II.

Physicochemical Properties

M.Wt	470.53
Formula	C23H28F2N8O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	[(S)-2-(1-(6-(((6,7-difluoro-1H-benzo[d]imidazol-2-yl)methyl)amino)-9-isopropyl-9H-purin-2-yl)piperidin-2-yl)ethan-1-ol]

References

1. Johannes JW, et al. ChemMedChem. 2018 Feb 6;13(3):231-235.

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CDK12-IN-3

Biological Activity

Physicochemical Properties

References

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