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Chemical Structure : CFI-401870
Catalog No.: PC-60266Not For Human Use, Lab Use Only.
CFI-401870 is a potent, selective, orally active Mps1 (TTK) inhibitor with IC50 of 3.1 nM.
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CFI-401870 is a potent, selective, orally active Mps1 (TTK) inhibitor with IC50 of 3.1 nM.
CFI-401870 displays low off-target activity (>500-fold) and microsomal stability.
CFI-401870 inhibits HCT116 cell growth with GI50 of <0.1 uM, demonstrates in vivo tumor growth inhibition.
| M.Wt | 493.611 | |
| Formula | C30H31N5O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Liu Y, et al. J Med Chem. 2015 Apr 23;58(8):3366-92.
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