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Chemical Structure : CH5447240
Catalog No.: PC-35255Not For Human Use, Lab Use Only.
CH5447240 is a novel potent, selective, orally active hPTHR1 agonist with EC20 of 3.0 nM and EC50 of 12 nM.
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CH5447240 is a novel potent, selective, orally active hPTHR1 agonist with EC20 of 3.0 nM and EC50 of 12 nM; shows excellent physicochemical properties, such as high solubility in fasted state simulated intestinal fluid and good metabolic stability in human liver microsomes; demonstrates a significantly elevated serum calcium level in hypocalcemic model rats.
| M.Wt | 517.689 | |
| Formula | C26H39N5O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Nishimura Y, et al. J Med Chem. 2018 Jun 22. doi: 10.1021/acs.jmedchem.8b00182.
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