Chemical Structure : CTAP
CAS No.: 103429-32-9
Catalog No.: PC-27170Not For Human Use, Lab Use Only.
CTAP is a potent, highly selective, and BBB-penetrant μ opioid receptor (MOR) antagonist with IC50 of 3.5 nM ,> 1200-fold selectivity over δ opioid receptor ( MOR, IC50=4500 nM) and somatostatin receptors.
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CTAP is a potent, highly selective, and BBB-penetrant μ opioid receptor (MOR) antagonist with IC50 of 3.5 nM ,> 1200-fold selectivity over δ opioid receptor ( MOR, IC50=4500 nM) and somatostatin receptors.
| M.Wt | 1104.30 | |
| Formula | C51H69N13O11S2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
{d-Phe}-Cys-Tyr-{d-Trp}-Arg-Thr-{Pen}-Thr-NH2 (Disulfide bridge:Cys2-Pen7) |
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1. Abbruscato TJ, et al. J Pharmacol Exp Ther. 1997 Jan;280(1):402-9.

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