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Chemical Structure : CV-6209
Catalog No.: PC-60754Not For Human Use, Lab Use Only.
A highly potent, selective platelet activating factor (PAF) inhibitor with IC50 of 75 and 170 nM for aggregation inhibition of rabbit and human platelets induced by PAF.
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A highly potent, selective platelet activating factor (PAF) inhibitor with IC50 of 75 and 170 nM for aggregation inhibition of rabbit and human platelets induced by PAF; shows little to no effects on the aggregation induced by arachidonic acid, ADP and collagen; inhibited PAF-induced hypotension in rats (ED50=0.009 mg/kg i.v.) with no effect on the hypotension induced by arachidonic acid, histamine, bradykinin and isoproterenol.
Ulcer
Discontinued
| M.Wt | 642.3 | |
| Formula | C34H60N3O6Cl | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Terashita Z, et al. J Pharmacol Exp Ther. 1987 Jul;242(1):263-8.
2. Terashita Z, et al. J Cardiovasc Pharmacol. 1988;12(5):505-11.
3. Stahl GL, et al. J Pharmacol Exp Ther. 1988 Mar;244(3):898-904.
4. Takatani M, et al. J Med Chem. 1989 Jan;32(1):56-64.
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