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CaSR-IN-10a

Chemical Structure : CaSR-IN-10a

CAS No.: 478963-79-0

CaSR-IN-10a (2(1H)-Quinazolinone, 1-(1-methylethyl)-4-[4-(1-methylethyl)phenyl]-6-(2-propyn-1-yloxy)-)

Catalog No.: PC-45852Not For Human Use, Lab Use Only.

A potent CaSR antagonist with IC50 of 4.4 nM in CaSR FLIPR assay..

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

A potent CaSR antagonist with IC50 of 4.4 nM in CaSR FLIPR assay.

Physicochemical Properties

M.Wt 360.4489
Formula C23H24N2O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

2(1H)-Quinazolinone, 1-(1-methylethyl)-4-[4-(1-methylethyl)phenyl]-6-(2-propyn-1-yloxy)-

References

1. Widler L, et al. J Med Chem. 2010 Mar 11;53(5):2250-63.

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