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Chemical Structure : Casopitant
Catalog No.: PC-61580Not For Human Use, Lab Use Only.
Casopitant (GW679769) is a potent, centrally-acting neurokinin 1 (NK1) receptor antagonist (pKi=9.48) with antidepressant and antiemetic activities.
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Casopitant (GW679769) is a potent, centrally-acting neurokinin 1 (NK1) receptor antagonist (pKi=9.48) with antidepressant and antiemetic activities; demonstrates potential for treatment of chemotherapy-induced nausea and vomiting (CINV).
Chemotherapeutic Agents
Phase 2 Discontinued
| M.Wt | 616.625 | |
| Formula | C30H35F7N4O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Minthorn E, et al. Drug Metab Dispos. 2008 Sep;36(9):1846-52.
2. Ruhlmann C, et al. Ther Clin Risk Manag. 2009 Apr;5(2):375-84.
3. Singla NK, et al. Anesthesiology. 2010 Jul;113(1):74-82.
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