D2AAK1

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Chemical Structure : D2AAK1

Catalog No.: PC-27970Not For Human Use, Lab Use Only.

D2AAK1 is a high-affinity dopamine D2 receptor antagonist with Ki of 58 nM, also possesses additional nanomolar or low micromolar affinity to D1, D3, 5-HT1A and 5-HT2A receptors, shows antipsychotic activity in vivo.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

D2AAK1 is a high-affinity dopamine D2 receptor antagonist with Ki of 58 nM, also possesses additional nanomolar or low micromolar affinity to D1, D3, 5-HT1A and 5-HT2A receptors, shows antipsychotic activity in vivo.

Physicochemical Properties

M.Wt	385.47
Formula	C24H23N3O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	3-((4-(5-methoxy-1H-indol-3-yl)-3,6-dihydropyridin-1(2H)-yl)methyl)quinolin-2(1H)-one

References

1. Kaczor AA, et al. Neurochem Int. 2016 Jun;96:84-99.

2. Koszła O, et al. Int J Mol Sci. 2020 Nov 23;21(22):8849.

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D2AAK1

Biological Activity

Physicochemical Properties

References

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