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DC591053

Chemical Structure : DC591053

CAS No.:

DC591053 (DC 591053)

Catalog No.: PC-20022Not For Human Use, Lab Use Only.

DC591053 (DC 591053) is a selective small molecule agonist of relaxin family peptide receptor 4 (RXFP4) with pEC50  of 7.24  and pKi  of  6.95, shows no activity against RXFP3.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

DC591053 (DC 591053) is a selective small molecule agonist of relaxin family peptide receptor 4 (RXFP4) with pEC50  of 7.24  and pKi  of  6.95, shows no activity against RXFP3.

Physicochemical Properties

M.Wt 493.60
Formula C28H35N3O5
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(S)-(7-ethoxy-6-methoxy-1-(2-(5-methoxy-1H-indol-3-yl)ethyl)-3,4-dihydroisoquinolin-2(1H)-yl)(morpholino)methanone

References

1. Yan Chen, et al. Nat Commun. 2023 Jan 30;14(1):492.

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