You are here:Home-Chemical Inhibitors & Agonists-GPCR-Opioid Receptor-DPI-287
DPI-287

Chemical Structure : DPI-287

CAS No.: 519058-13-0

DPI-287 (DPI 287)

Catalog No.: PC-49552Not For Human Use, Lab Use Only.

DPI-287 is a small-molecule agonist of the δ-opioid receptor (DOP) with Ki vaule of 0.39 nM, shows 10-fold selectivity for DOP over MOP (Ki=3.17 nM).

Packing Price Stock Quantity
100 mg Get quote
250 mg Get quote
500 mg Get quote
1 g Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC)

Biological Activity

DPI-287 is a small-molecule agonist of the δ-opioid receptor (DOP) with Ki vaule of 0.39 nM, shows 10-fold selectivity for DOP over MOP (Ki=3.17 nM).

Physicochemical Properties

M.Wt 485.67
Formula C31H39N3O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

4-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)-N,N-diethylbenzamide

References

1. Tobias Claff, et al. Sci Adv. 2019 Nov 27;5(11):eaax9115.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: