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DRAK2 inhibitor 16

Chemical Structure : DRAK2 inhibitor 16

CAS No.: 871837-60-4

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DRAK2 inhibitor 16 (DRAK2-IN-1)

Catalog No.: PC-62719Not For Human Use, Lab Use Only.

DRAK2 inhibitor 16 (DRAK2-IN-1) is a potent, selective DRAK2 (STK17B) inhibitor with IC50 of 3 nM, shows weaker inhibition for DRAK1 (IC50=51 nM) and no significant activity against DAPK1/2/3 (IC50>1 uM).

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

DRAK2 inhibitor 16 (DRAK2-IN-1) is a potent, selective DRAK2 (STK17B) inhibitor with IC50 of 3 nM, shows weaker inhibition for DRAK1 (IC50=51 nM) and no significant activity against DAPK1/2/3 (IC50>1 uM).

Physicochemical Properties

M.Wt 376.416
Formula C21H20N4O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-((2Z,3E)-3-(hydroxyimino)-2'-oxo-[2,3'-biindolinylidene]-5'-yl)pentanamide

References

1. Jung ME, et al. Bioorg Med Chem Lett. 2016 Jun 1;26(11):2719-23.

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