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Chemical Structure : DS-6930
Catalog No.: PC-35674Not For Human Use, Lab Use Only.
DS-6930 (DS 6930, DS6930) is a novel potent, selective PPARγ agonist with EC50 of 41 nM, Emax-68%.
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DS-6930 (DS 6930, DS6930) is a novel potent, selective PPARγ agonist with EC50 of 41 nM, Emax-68%; significantly recruits several cofactors, such as RIP140 and PGC1, in cofactor recruitment assays; demonstrateshigh PPARγ agonist potency with robust plasma glucose reduction, maintains diminished PPARγ-related adverse effects upon toxicological evaluation in vivo, and demonstrated no hepatotoxicity.
Diabetes
Discontinued
| M.Wt | 403.438 | |
| Formula | C23H21N3O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Shinozuka T, et al. Bioorg Med Chem. 2018 Oct 1;26(18):5099-5117.
2. Shinozuka T, et al. Bioorg Med Chem. 2018 Oct 1;26(18):5079-5098.
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