Chemical Structure : ENMD-2076
CAS No.: 934353-76-1
Catalog No.: PC-42766Not For Human Use, Lab Use Only.
A multitargeted kinase inhibitor with IC50s of 3/14/23/40 nM for Flt3/Aurora A/Src/VEGFR2.
Packing | Price | Stock | Quantity |
---|---|---|---|
10 mg | $120 | In stock | |
50 mg | $360 | In stock | |
100 mg | $520 | In stock |
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
A multitargeted kinase inhibitor with IC50s of 3/14/23/40 nM for Flt3/Aurora A/Src/VEGFR2; also inhibits Aurora B, c-Kit, FGFR1 (IC50=100-350 nM); orally bioactive.
M.Wt | 375.4701 | |
Formula | C21H25N7 | |
Appearance | Solid | |
Storage |
|
|
Solubility |
10 mM in DMSO |
|
Chemical Name/SMILES |
4-Pyrimidinamine, 6-(4-methyl-1-piperazinyl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(1E)-2-phenylethenyl]- |
1. Tentler JJ, et al. Clin Cancer Res. 2010 Jun 1;16(11):2989-98.
2. Matulonis UA, et al. Eur J Cancer. 2013 Jan;49(1):121-31.
3. Fletcher GC, et al. Mol Cancer Ther. 2011 Jan;10(1):126-37.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright