ENMD-2076 tartrate | Multikinase inhibitor

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Chemical Structure : ENMD-2076 tartrate

CAS No.: 1291074-87-7

ENMD-2076 tartrate (ENMD 2076, ENMD2076)

Catalog No.: PC-42765Not For Human Use, Lab Use Only.

ENMD-2076 tartrate is a multitargeted kinase inhibitor with IC50s of 3/14/23/40 nM for Flt3/Aurora A/Src/VEGFR2; also inhibits Aurora B, c-Kit, FGFR1 (IC50=100-350 nM); orally bioactive.

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25 mg	$138	In stock
50 mg	$218	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

ENMD-2076 tartrate is a multitargeted kinase inhibitor with IC50s of 3/14/23/40 nM for Flt3/Aurora A/Src/VEGFR2; also inhibits Aurora B, c-Kit, FGFR1 (IC50=100-350 nM); orally bioactive.

Physicochemical Properties

M.Wt	525.5569
Formula	C25H31N7O6
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	4-Pyrimidinamine, 6-(4-methyl-1-piperazinyl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(1E)-2-phenylethenyl]- Tartrate

References

1. Tentler JJ, et al. Clin Cancer Res. 2010 Jun 1;16(11):2989-98.

2. Matulonis UA, et al. Eur J Cancer. 2013 Jan;49(1):121-31.

3. Fletcher GC, et al. Mol Cancer Ther. 2011 Jan;10(1):126-37.

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ENMD-2076 tartrate (ENMD 2076, ENMD2076)

Biological Activity

Physicochemical Properties

References

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