You are here:Home-Chemical Inhibitors & Agonists-GPCR-P2Y Receptor-Elinogrel
Elinogrel

Chemical Structure : Elinogrel

CAS No.: 936500-94-6

Elinogrel (PRT-060128;PRT060128)

Catalog No.: PC-61587Not For Human Use, Lab Use Only.

Elinogrel (PRT060128) is a selective, reversible, competitive and direct-acting P2Y12 receptor antagonist for the treatment of acute coronary syndrome and prevention of secondary thrombotic events..

Packing Price Stock Quantity

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Elinogrel (PRT060128) is a selective, reversible, competitive and direct-acting P2Y12 receptor antagonist for the treatment of acute coronary syndrome and prevention of secondary thrombotic events.

Thrombosis

Phase 2 Discontinued

Physicochemical Properties

M.Wt 523.945
Formula C20H15ClFN5O5S2
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-[4-(6-Fluoro-7-methylamino-2,4-dioxo-1,4-dihydro-2H-quinazolin-3-yl)phenyl]-N'-[(5-chlorothiophen-2-yl)sulfonyl]urea

References

1. Siller-Matula JM, et al. Br J Pharmacol. 2010 Feb 1;159(3):502-17.

2. Leonardi S, et al. Am Heart J. 2010 Jul;160(1):65-72.

3. Oestreich JH. Curr Opin Investig Drugs. 2010 Mar;11(3):340-8.

4. André P, et al. J Pharmacol Exp Ther. 2011 Jul;338(1):22-30.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: