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Chemical Structure : G-9791
Catalog No.: PC-60221Not For Human Use, Lab Use Only.
G-9791 (G9791) is a potent and selective group I PAK (pan-PAK1/2/3) inhibitor with Ki of 0.95/2 nM for PAK1/2, respectively.
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G-9791 (G9791) is a potent and selective group I PAK (pan-PAK1/2/3) inhibitor with Ki of 0.95/2 nM for PAK1/2, respectively.
G-9791 displays 57-fold selectivity over Lck kinase.
G-9791 inhibits the phosphorylation of residue S298 of MEK1 in EBC1 cells with IC50 of 33 nM.
| M.Wt | 508.98 | |
| Formula | C26H26ClFN6O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Rudolph J, et al. J Med Chem. 2016 Jun 9;59(11):5520-41.
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