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GK442

Chemical Structure : GK442

CAS No.: 2047917-85-9

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GK442 (GK-442)

Catalog No.: PC-23707Not For Human Use, Lab Use Only.

GK442 is a highly potent autotaxin inhibitor with IC50 of 60 nM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

GK442 is a highly potent autotaxin inhibitor with IC50 of 60 nM.
GK442 (30 mg/kg, i.p.) exhibited promising efficacy in a mouse model of pulmonary inflammation and fibrosis induced by bleomycin.

Physicochemical Properties

M.Wt 391.51
Formula C21H33N3O4
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(S)-N1-(1-(Hydroxyamino)-1-oxononan-5-yl)-N6-phenyladipamide

References

1. Nikolaou A, et al. J Med Chem. 2018 Apr 26;61(8):3697-3711.

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