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GPR4 antagonist 39c

Chemical Structure : GPR4 antagonist 39c

CAS No.: 1197879-16-5

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GPR4 antagonist 39c

Catalog No.: PC-20836Not For Human Use, Lab Use Only.

GPR4 antagonist 39c is a potent and orally active GPR4 antagonist with IC50 of 110 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    GPR4 antagonist 39c is a potent and orally active GPR4 antagonist with IC50 of 110 nM.
    GPR4 antagonist 39c shows potent cellular activity and is efficacious in animal models of angiogenesis, inflammation and pain.

    Physicochemical Properties

    M.Wt 431.63
    Formula C27H37N5
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (E)-2-ethyl-3-(4-(3-(4-isopropylpiperazin-1-yl)prop-1-en-1-yl)benzyl)-5,7-dimethyl-3H-imidazo[4,5-b]pyridine

    References

    1. Wolfgang Miltz, et al. Bioorg Med Chem. 2017 Aug 15;25(16):4512-4525.

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