You are here:Home-Chemical Inhibitors & Agonists-GPCR-Proton-sensing GPCRs-GPR4 antagonist 39c
GPR4 antagonist 39c

Chemical Structure : GPR4 antagonist 39c

CAS No.: 1197879-16-5

GPR4 antagonist 39c

Catalog No.: PC-20836Not For Human Use, Lab Use Only.

GPR4 antagonist 39c is a potent and orally active GPR4 antagonist with IC50 of 110 nM.

Packing Price Stock Quantity
25 mg Get quote
100 mg Get quote
200 mg Get quote
1 g Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC)

Biological Activity

GPR4 antagonist 39c is a potent and orally active GPR4 antagonist with IC50 of 110 nM.
GPR4 antagonist 39c shows potent cellular activity and is efficacious in animal models of angiogenesis, inflammation and pain.

Physicochemical Properties

M.Wt 431.63
Formula C27H37N5
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

CC1=C2C(N(CC3=CC=C(/C=C/CN4CCN(C(C)C)CC4)C=C3)C(CC)=N2)=NC(C)=C1

References

1. Wolfgang Miltz, et al. Bioorg Med Chem. 2017 Aug 15;25(16):4512-4525.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: