GR128107 | Melatonin receptor antagonist

Chemical Structure : GR128107

GR128107 (GR 128107, GR-128107)

Catalog No.: PC-26839Not For Human Use, Lab Use Only.

GR128107 is a high affinity, competitive melatonin receptor antagonist with pKi of 9.6, shows substantially higher affinities for MT2 receptor, 23 fold selective over MT1.

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Biological Activity

GR128107 is a high affinity, competitive melatonin receptor antagonist with pKi of 9.6, shows substantially higher affinities for MT2 receptor, 23 fold selective over MT1.

Physicochemical Properties

M.Wt	272.35
Formula	C16H20N2O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(3-(5-methoxy-1H-indol-3-yl)piperidin-1-yl)ethan-1-one

References

1. Dubocovich ML, et al. Naunyn Schmiedebergs Arch Pharmacol. 1997 Mar;355(3):365-75.

2. Teh MT, et al. Br J Pharmacol. 1999 Mar;126(5):1237-45.

3. Browning C, et al. Br J Pharmacol. 2000 Mar;129(5):877-86.

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GR128107 (GR 128107, GR-128107)

Biological Activity

Physicochemical Properties

References

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