Catalog No.: PC-26007Not For Human Use, Lab Use Only.
GSK1362 (GSK3201362) is a specific small molecule ligand with inverse agonist properties of REV-ERB, disrupts the interaction of REV-ERBα with repressive co-modulators (NCoR1, SMRT2, RIP140), demonstrates upregulation of BMAL1 gene transcription with EC50 of 2.5 uM.
GSK1362 (GSK3201362) is a specific small molecule ligand with inverse agonist properties of REV-ERB, disrupts the interaction of REV-ERBα with repressive co-modulators (NCoR1, SMRT2, RIP140), demonstrates upregulation of BMAL1 gene transcription with EC50 of 2.5 uM.
